O PCE 10mg Pellets – Advanced Research Formulation for Neuropsychopharmacology
O PCE
🔬Especificações técnicas
IUPAC Name: 2-(Ethylamino)-2-(2-methoxyphenyl)cyclohexan-1-one
Alternative Name: 2′-Oxo-PCE
Dosagem: 10mg ± 0.2mg per pellet (pharmaceutical precision)
Forma: Round, uniform pellets (Ø 5mm)
Cor: Light beige (natural dye)
Tempo de desintegração: <15 minutes (USP method)
Coating: Vegetarian HPMC film coating
🧠Neuroscience Applications
✔ NMDA receptor modulation studies
✔ Neuroprotective mechanisms research
✔ Non-animal in vitro models
✔ Comparative pharmacokinetics
⚗️Garantias de qualidade
Produção com certificação GMP
Triplo controlo de qualidade:
UHPLC-PDA (purity ≥98.5%)
GC-MS (residual solvents <50ppm)
Karl Fischer (moisture content <0.5%)
Dados de estabilidade: 24 months under conditioned storage
☢️Safety protocol
Biosafety Level 2 required
EPI obrigatório:
Luvas de nitrilo (sem talco)
Máscara facial tipo IIR
Closed system transfer
Spill procedure:
Absorbent polymer + 5% acetic acid solution
🌡️Storage matrix
| Packaging level | Material | O2 barrier | Moisture control |
|---|---|---|---|
| Primary | Alu-alu blister | <0.1% O2 | Silica gel |
| Secondary | Amber silica pot | <0.5% O2 | Desiccant |
📊Dosage accuracy
Batch # | Average (mg) | RSD (%) | N=30 OPCE-2401 | 10.05 | 0.9% OPCE-2402 | 9.98 | 1.1%
⚖️Regulatory Framework
Dutch Opium Act Special Category
EU NPS Monitoring System
Export control:
DEA Form 486 required
End-Use Declaration mandatory
🔍Apoio analítico
Included as standard:
Chirality analysis (HPLC-CD)
DSC thermogram
Premium options:
In vitro blood-brain barrier permeability
Microsome stability studies
🚨Ethical Guidelines:
This formulation is exclusively intended for:
Certified research institutions
Pharmaceutical development laboratories
📚Academic Collaboration:
We support:
In silico receptor docking studies
Structural modification research
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